Final published version
Research output: Contribution to Journal/Magazine › Journal article › peer-review
| <mark>Journal publication date</mark> | 1/09/1993 |
|---|---|
| <mark>Journal</mark> | SYNLETT |
| Issue number | 9 |
| Volume | 1993 |
| Number of pages | 2 |
| Pages (from-to) | 675-676 |
| Publication Status | Published |
| <mark>Original language</mark> | English |
The novel ring-opening reaction of enantiopure N-activated aziridines 1 with anions 2 derived from 1,3-dithiane proceeds regiospecifically at the carbon of lesser substitution. The ring-opened products 3 may efficiently be converted to homochiral 2-tosylaminocarbonyl compounds 4.