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Ring-opening of N-tosyl aziridines by sulphur-stabilized nucleophiles

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<mark>Journal publication date</mark>1/09/1993
<mark>Journal</mark>SYNLETT
Issue number9
Volume1993
Number of pages2
Pages (from-to)675-676
Publication StatusPublished
<mark>Original language</mark>English

Abstract

The novel ring-opening reaction of enantiopure N-activated aziridines 1 with anions 2 derived from 1,3-dithiane proceeds regiospecifically at the carbon of lesser substitution. The ring-opened products 3 may efficiently be converted to homochiral 2-tosylaminocarbonyl compounds 4.