Final published version
Research output: Contribution to Journal/Magazine › Journal article › peer-review
Research output: Contribution to Journal/Magazine › Journal article › peer-review
}
TY - JOUR
T1 - Ring-opening of N-tosyl aziridines by sulphur-stabilized nucleophiles
AU - Osborn, Helen M.I.
AU - Sweeney, J. B.
AU - Howson, Bill
PY - 1993/9/1
Y1 - 1993/9/1
N2 - The novel ring-opening reaction of enantiopure N-activated aziridines 1 with anions 2 derived from 1,3-dithiane proceeds regiospecifically at the carbon of lesser substitution. The ring-opened products 3 may efficiently be converted to homochiral 2-tosylaminocarbonyl compounds 4.
AB - The novel ring-opening reaction of enantiopure N-activated aziridines 1 with anions 2 derived from 1,3-dithiane proceeds regiospecifically at the carbon of lesser substitution. The ring-opened products 3 may efficiently be converted to homochiral 2-tosylaminocarbonyl compounds 4.
U2 - 10.1055/s-1993-22568
DO - 10.1055/s-1993-22568
M3 - Journal article
AN - SCOPUS:0002145831
VL - 1993
SP - 675
EP - 676
JO - SYNLETT
JF - SYNLETT
SN - 0936-5214
IS - 9
ER -